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Monograph
RESEARCH GREYP-018
Recovery

Larazotide

Octapeptide tight-junction regulator. Antagonizes zonulin to restore intestinal epithelial barrier integrity.

EmergingRecovery
Typical dose0.5 mg
Frequencybefore meals, oral
Half-life0.5h
Citations indexed27
DeliveryInjectable
Half-life~30min
EvidenceEmerging
Citations27
Synergy checkCompareReconstitution calc
Research grey

This compound sits in research-grey territory. The caveats below carry more weight than for FDA-approved entries — read them.

Mechanism

9 Meters Biopharma's lead candidate (CEDLARA Phase 3 in celiac). Reduces tight-junction permeability rather than directly modulating immune cells. Phase 3 results were mixed in 2022. Still positioned as an adjunct for refractory celiac and explored for long-COVID gut symptoms.

Specifics
Slow wound healing
Caveats

Not approved. Phase 3 results were not unambiguously positive. Self-experimentation outside trial protocols carries unknown long-term risk for chronic GI conditions.

sequence · 8 aa
GGVLVQPG
Evidence levelEmerging
Regulatory statusInvestigational — phase 3 celiac results mixed 2022
DNA / pharmacogenomicsLow — HLA-DQ2/DQ8 status matters for celiac diagnosis, not response to larazotide.
Claims & evidence

Per-claim grading. Each claim is graded independently — same peptide, different claims can carry different grades.

  • CLimited evidence

    Larazotide — primary mechanism: octapeptide tight-junction regulator. antagonizes zonulin to restore intestinal epithelial barrier integrity.

    2 supporting referencesVerified 5d ago
References

External links to PubMed searches, ClinicalTrials.gov, and FDA materials. We do not host papers — we point at canonical sources.

  • PubMedEN
    REVIEWFunding undisclosedVerified 5d ago
    PubMed — Larazotide celiac
  • Clinical trialEN
    RCTFunding undisclosedVerified 5d ago
    ClinicalTrials.gov — CEDLARA
Reconstitution calculatorLarazotide

Pre-filled with this compound's published dose range: 0.5 mg · before meals, oral

Concentration2.50 mg/mL
Draw volume0.200 mL
Insulin syringe20.0 u
Doses per vial10
U-100 syringe — fill to indicatorU-100 · 1 mL
0u25u50u75u100u

Calculator is a discussion tool. Verify reconstitution + dosing with a qualified provider. Stack is not a prescription source. Use sterile technique and inspect every vial.

RESEARCH GREYP-018

Investigational — phase 3 celiac results mixed 2022

Larazotide0.5 mg · before meals, oral
Discussion guide, not prescription

stack is an exploration engine. Output is a discussion guide for a conversation with a licensed provider — never a prescription, dose recommendation, or sourcing instruction. Peptides discussed include compounds with limited human evidence and varying legal status by jurisdiction. Verify everything with a qualified clinician before any decision.

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